A new route to 5-aryl and 5-heteroaryl-2-pyrones via Suzuki coupling of a 2-pyrone-5-boronate ester

Edward C. Gravett; Philip J. Hilton; Keith Jones; Jean Marie Péron

doi:10.1055/s-2003-36789

A new route to 5-aryl and 5-heteroaryl-2-pyrones via Suzuki coupling of a 2-pyrone-5-boronate ester

Edward C. Gravett
, Philip J. Hilton
, Keith Jones
, Jean Marie Péron

Research output: Contribution to journal › Article › peer-review

Abstract

A synthesis of boronate (III) is reported along with its use in Pd-catalyzed coupling reactions with aryl halides and triflates. Catalytic hydrogenation of the resulting products provides a rapid way of introducing a valerolactone residue onto an aromatic ring.

Original language	English
Pages (from-to)	0253-0255
Journal	Synlett
Volume	2
DOIs	https://doi.org/10.1055/s-2003-36789
Publication status	Published - Feb 2003

Keywords

Suzuki coupling
palladium
boron
heterocycles
pyrone
radicals
Chemistry

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10.1055/s-2003-36789

http://dx.doi.org/10.1055/s-2003-36789

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title = "A new route to 5-aryl and 5-heteroaryl-2-pyrones via Suzuki coupling of a 2-pyrone-5-boronate ester",

abstract = "A synthesis of boronate (III) is reported along with its use in Pd-catalyzed coupling reactions with aryl halides and triflates. Catalytic hydrogenation of the resulting products provides a rapid way of introducing a valerolactone residue onto an aromatic ring.",

keywords = "Suzuki coupling, palladium, boron, heterocycles, pyrone, radicals, Chemistry",

author = "Gravett, \{Edward C.\} and Hilton, \{Philip J.\} and Keith Jones and P{\'e}ron, \{Jean Marie\}",

year = "2003",

month = feb,

doi = "10.1055/s-2003-36789",

language = "English",

volume = "2",

pages = "0253--0255",

journal = "Synlett",

issn = "0936-5214",

publisher = "Georg Thieme Verlag",

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T1 - A new route to 5-aryl and 5-heteroaryl-2-pyrones via Suzuki coupling of a 2-pyrone-5-boronate ester

AU - Gravett, Edward C.

AU - Hilton, Philip J.

AU - Jones, Keith

AU - Péron, Jean Marie

PY - 2003/2

Y1 - 2003/2

N2 - A synthesis of boronate (III) is reported along with its use in Pd-catalyzed coupling reactions with aryl halides and triflates. Catalytic hydrogenation of the resulting products provides a rapid way of introducing a valerolactone residue onto an aromatic ring.

AB - A synthesis of boronate (III) is reported along with its use in Pd-catalyzed coupling reactions with aryl halides and triflates. Catalytic hydrogenation of the resulting products provides a rapid way of introducing a valerolactone residue onto an aromatic ring.

KW - Suzuki coupling

KW - palladium

KW - boron

KW - heterocycles

KW - pyrone

KW - radicals

KW - Chemistry

U2 - 10.1055/s-2003-36789

DO - 10.1055/s-2003-36789

M3 - Article

SN - 0936-5214

VL - 2

SP - 253

EP - 255

JO - Synlett

JF - Synlett

ER -

A new route to 5-aryl and 5-heteroaryl-2-pyrones via Suzuki coupling of a 2-pyrone-5-boronate ester

Abstract

Keywords

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