An expedient conversion of [alpha]-amino acids into Weinreb amides using COMU (R) as a coupling agent

  • Elizabeth Tyrrell
  • , Peter Brawn
  • , Mark Carew
  • , Iain Greenwood

    Research output: Contribution to journalArticlepeer-review

    Original languageEnglish
    Pages (from-to)369-372
    JournalTetrahedron Letters
    Volume52
    Issue number3
    DOIs
    Publication statusPublished - Jan 2011

    Keywords

    • weinreb amides
    • calorimetric changes
    • amidation
    • water-soluble by-products
    • comu (r)
    • methoxy-n-methylamides
    • effective acylating agents
    • asymmetric-synthesis
    • enantioselective synthesis
    • peptide-synthesis
    • ketones
    • route
    • construction
    • equivalents
    • derivatives
    • Pharmacy

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